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名称

Endomorphin 2 TFA

别名

内吗啡肽2TFA

英文名称

Endomorphin 2 TFA

货号

E650113-5mg

包装规格

5mg

浓度

≥99%

储存温度

干燥,-80℃储存

运输条件

超低温冰袋运输

产品介绍

Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor , displays reasonable affinities for kappa 3 binding sites, with K i value between 20 and 30 nM Form:Solid IC50& Target:Ki: 20-30 nM (kappa 3 opioid receptor)

生化机理

Endomorphin 2 TFA 是一种高亲和力、高选择性的μ-阿片受体激动剂，对 kappa 3 结合位点具有合理的亲和力，其 K i 值介于 20 至 30 nM 之间。

CAS号

1276124-00-5

分子式

C34H38F3N5O7

分子量

685.69 g/mol

PubChem编号

137700452

IIUPAC Name

(2S)-1-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]-N-[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]pyrrolidine-2-carboxamide;2,2,2-trifluoroacetic acid

INCHI

1S/C32H37N5O5.C2HF3O2/c33-25(18-23-13-15-24(38)16-14-23)32(42)37-17-7-12-28(37)31(41)36-27(20-22-10-5-2-6-11-22)30(40)35-26(29(34)39)19-21-8-3-1-4-9-21;3-2(4,5)1(6)7/h1-6,8-11,13-16,25-28,38H,7,12,17-20,33H2,(H2,34,39)(H,35,40)(H,36,41);(H,6,7)/t25-,26-,27-,28-;/m0./s1

InChi Key

ONJAQAAWBPIPNC-ZLYCMTQRSA-N

Smiles

C1CC(N(C1)C(=O)C(CC2=CC=C(C=C2)O)N)C(=O)NC(CC3=CC=CC=C3)C(=O)NC(CC4=CC=CC=C4)C(=O)N.C(=O)(C(F)(F)F)O

PubChem CID

137700452

溶解性

H2O : 62.5 mg/mL (91.15 mM; Need ultrasonic) DMSO : 6 mg/mL (8.75 mM; Need ultrasonic)

Safety

「No Dangerous Attributes」

「No upstream and downstream information yet」

Technical Documents

「No technical documents」

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「No related articles yet」

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