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Product introduction

EN219 is a moderately selective synthetic covalent ligand against an N-terminal cysteine (C8) of RNF114 with an IC 50 of 470 nM. EN219 inhibits RNF114-mediated autoubiquitination and p21 ubiquitination In Vitro EN219 (1 μM; 90 min) interacts with RNF114 C8, TUBB1 C201, HSPD1 C442, and HIST1H3A C97 demonstrated by isotopic tandem orthogonal proteolysisABPP (isoTOP-ABPP) analysis. MCE has not independently confirmed the accuracy of these methods. They are for reference only. Form:Solid IC50& Target:RNF114 470 nM (IC 50 )

Specs ⸢ View details ⸥

Chinese name

EN219

English name

EN219

Chinese alias

English alias

CAS number

380351-29-1

molecular formula

C17H13Br2ClN2O

molecular weight

456.56 g/mol

Exact mass

≥98%

PSA

Logp

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