Share to

Overview

Specs

Technical Documents

Articles

reviews

Consult

returns

Product introduction

GNE-0439 is a novel Nav1.7 -selective inhibitor with IC 50 of 0.34 uM and inhibits Nav1.5 with an IC 50 of 38.3 μM. GNE-0439 inhibits mutant N1742K channels ( IC 50 =0.37 uM) in membrane potential assays. GNE-0439 possesses a carboxylic acid group, binds outside of the channel pore, and is unique compared with known selective VSD4 binders Form:Solid IC50& Target:IC50: 0.34 uM (Nav1.7)

Specs ⸢ View details ⸥

Chinese name

GNE-0439

English name

GNE-0439

Chinese alias

English alias

CAS number

1241902-40-8

molecular formula

C21H31NO3

molecular weight

345.48 g/mol

Exact mass

≥99%

PSA

Logp

Technical Documents

「No technical documents」

「No upstream and downstream information yet」

Articles

「No related articles yet」

user reviews

Consultation

Warm reminder：

Because the manufacturer may temporarily adjust product specifications, prices, inventory, parameters and other information without notice, and there are differences in each user's consultation time and procurement needs, the platform reply content is only of reference value within a certain period. Sorry for the inconvenience caused to you, and thank you for your understanding and support! Please consult the online customer service for the latest details. Everything is subject to the real-time reply of the customer service.！

After Sales Services

Please check the quantity, appearance and product information in time when you receive the goods. In case of damage, wrong delivery, abnormal quality and other problems, please feel free to contact us.

Service Hotline:400-6226-992 ，We will handle it for you as soon as possible, thank you for your support and trust.！