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Product introduction

Peficitinib (ASP015K, JNJ-54781532)是一种口服具有生物活性的 JAK 抑制剂。 Information Peficitinib (ASP015K, JNJ-54781532) is an orally bioavailableJAKinhibitor. Phase 3. Targets JAK In vitro ASP015K suppresses the IL-2-induced proliferation of human T cells with greater potency than EPO-induced proliferation of human erythroleukemia cells. In human whole blood, ASP015K inhibits STAT5 phosphorylation (pSTAT5). In vivo In the rat AIA model, ASP015K (p.o.) significantly decreases paw swelling and ankle bone destruction score.

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Chinese name

培菲替尼（ASP015K）, Janus 激酶 1 抑制剂

English name

Peficitinib (ASP015K)

Chinese alias

English alias

4-(((1R,2s,3S,5s,7s)-5-hydroxyadamantan-2-yl)amino)-1H-pyrrolo(2,3-b)pyridine-5-carboxamide | 1H-Pyrrolo(2,3-b)pyridine-5-carboxamide, 4-((5-hydroxytricyclo(3.3.1.13,7)dec-2-yl)amino)-, stereoisomer | GTPL8315 | AMY42225 | 9T6 | PEFICITINIB [INN] | JNJ-54

CAS number

944118-01-8

molecular formula

C18H22N4O2

molecular weight

326.39 g/mol

Exact mass

PSA

104.000 Å²

Logp

1.900

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Peficitinib (ASP015K, JNJ-54781532) 10mM in DMSO 1ml

Name: Peficitinib (ASP015K, JNJ-54781532) 10mM in DMSO 1ml
Brand: 麦克林
SKU: P797406-1ml

Peficitinib (ASP015K, JNJ-54781532) 10mM in DMSO 1ml Macklin 944118-01-8, complete specifications, for production, research, laboratory testing and inspection, digital one-stop procurement platform for scientific materials.

item number：P797406-1ml

Product model：1ml

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Lead Time：30days

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Peficitinib (ASP015K, JNJ-54781532) 10mM in DMSO 1ml

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