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Product details

名称

RF9 hydrochloride

别名

RF9 盐酸盐

英文名称

RF9 hydrochloride

货号

R658968-5mg

包装规格

5mg

浓度

≥99%

储存温度

-20°C储存,干燥

运输条件

超低温冰袋运输

产品介绍

RF9 hydrochloride is a potent and selective Neuropeptide FF receptor antagonist, with K i values of 58 and 75 nM for hNPFF1R and hNPFF2R , respectively. Appearance:Solid IC50& Target:hNPFF1R 58 nM (Ki) hNPFF2R 75 nM (Ki) In Vitro:RF9 (10 μM) pretrement completely blocks NPFF induced neurite outgrowth of Neuro 2A cells. MCE has not independently confirmed the accuracy of these methods. They are for reference only. In Vivo:RF9 (0.1mg/kg, s.c. ) with heroin coadministration prevents heroin-induced delayed hyperalgesia and tolerance. RF9 (10 μg) infused alone does not result in a significant alteration of MAP or heart rate. Conversely, MAP and heart rate increases evoke Biological Activity:RF9 hydrochloride is a potent and selective Neuropeptide FF receptor antagonist, with K i values of 58 and 75 nM for hNPFF1R and hNPFF2R , respectively .

分子式

C26H39ClN6O3

分子量

519.08 g/mol

Smiles

NC(C(CC1=CC=CC=C1)NC([C@H](CCCNC(N)=N)NC(C23C[C@H](C4)CC(C[C@@H]4C3)C2)=O)=O)=O.Cl

溶解性

DMSO : 50 mg/mL (96.32 mM; Need ultrasonic)

Safety

「No Dangerous Attributes」

「No upstream and downstream information yet」

Technical Documents

「No technical documents」

Articles

「No related articles yet」

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