Share to

Overview

Specs

Technical Documents

Articles

reviews

Consult

returns

Product introduction

Information TAK-063 (Balipodect) is a novel and selectivephosphodiesterase 10A(PDE10A)inhibitor with an IC50 of 0.30 nM. Targets PDE10A (Cell-free assay) 0.3 nM In vivo TAK-063 has high brain penetration in mice. Oral administration of TAK-063 to mice elevated striatal cAMP and (cGMP) levels at 0.3 mg/kg and shows potent suppression of phencyclidine (PCP)-induced hyperlocomotion at a minimum effective dose (MED) of 0.3 mg/kg. TAK-063 is currently being evaluated in clinical trials for the treatment of schizophrenia.

Specs ⸢ View details ⸥

Chinese name

TAK-063, 磷酸二酯酶 10A 抑制剂

English name

TAK-063

Chinese alias

English alias

HY-12472 | TAK063 | TAK-063 | BS-15045 | DB14774 | 1-(2-FLUORO-4-(1H-PYRAZOL-1-YL)PHENYL)-5-METHOXY- 3-(1-PHENYL-1H-PYRAZOL-5-YL)PYRIDAZIN-4(1H)-ONE | 3K9 | J-690093 | 1-[2-fluoro-4-(1H-pyrazol-1-yl)phenyl]-5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)-1,4-dihyd

CAS number

1238697-26-1

molecular formula

C23H17FN6O2

molecular weight

428.42 g/mol

Exact mass

10mM in DMSO

PSA

77.500 Å²

Logp

3.983

Technical Documents

「No technical documents」

「No upstream and downstream information yet」

Articles

「No related articles yet」

user reviews

Consultation

Warm reminder：

Because the manufacturer may temporarily adjust product specifications, prices, inventory, parameters and other information without notice, and there are differences in each user's consultation time and procurement needs, the platform reply content is only of reference value within a certain period. Sorry for the inconvenience caused to you, and thank you for your understanding and support! Please consult the online customer service for the latest details. Everything is subject to the real-time reply of the customer service.！

After Sales Services

Please check the quantity, appearance and product information in time when you receive the goods. In case of damage, wrong delivery, abnormal quality and other problems, please feel free to contact us.

Service Hotline:400-6226-992 ，We will handle it for you as soon as possible, thank you for your support and trust.！

MedMol TAK-063 98% 5mg

Name: MedMol TAK-063 98% 5mg
Brand: MedMol
SKU: S80213-5mg

MedMol TAK-063 98% 5mg, complete specifications; suitable for production, research, laboratory testing and inspection; digital one-stop procurement platform for scientific materials.

item number：S80213-5mg

Product model：5mg

level：

Lead Time：30days

sold 108 Items

Ask Solution engineer

Qty

MedMol TAK-063 98% 5mg

Recommended for you