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Product introduction

Trimipramine maleate 是 5-HT 受体的拮抗剂，其对 5-HT1C，5-HT2 和 5-HT1A 受体的 pKi 值分别为 6.39，8.10，4.66。Trimipramine maleate 也是一种靶向人去甲肾上腺素 (hNAT)、血清素 (hSERT) 和有机阳离子转运体 (hOCT1、hOCT2) 的有选择性和强效的抑制剂，其 IC50 值分别为 4.99 μM、2.11 μM、3.72 μM、8.00 μM。Trimipramine maleate 具有血管活性和抗焦虑作用。 Product description： Trimipramine maleate is a 5-HT receptor antagonist, with pKi binding values of 6.39, 8.10, 4.66 for 5-HT1C, 5-HT2 and 5-HT1A, respectively. Trimipramine maleate is also a potent and selective inhibitor targeting human noradrenaline (hNAT), serotonin (hSERT) and organic cation transporters (hOCT1, hOCT2) with IC50 values of 4.99 μM, 2.11 μM, 3.72 μM, 8.00 μM, respectively. Trimipramine maleate has vascular activity and anxiolytic efficacy.

Specs ⸢ View details ⸥

Chinese name

Trimipramine maleate salt, 肾上腺素能受体 alpha-1 拮抗剂

English name

Trimipramine maleate salt

Chinese alias

三甲丙咪嗪马来酸盐 | 马来酸三甲丙咪嗪 | 马来酸曲米帕明 | 马来酸曲米帕明

English alias

10,11-dihydro-N,N,beta-trimethyl-5H-dibenz(b,f)azepine-5-propanamine (Z)-2-butenedioate (1:1) | 5H-DIBENZ(B,F)AZEPINE-5-PROPANAMINE, 10,11-DIHYDRO-N,N,.BETA.-TRIMETHYL-, (Z)-2-BUTENEDIOATE (1:1) | 5H-DIBENZ(B,F)AZEPINE-5-PROPANAMINE, 10,11-DIHYDRO-N,N,.BE

CAS number

521-78-8

molecular formula

C24H30N2O4

molecular weight

410.51 g/mol

Exact mass

≥98%

PSA

81.100 Å²

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MedMol Trimipramine Maleate Salt 98% 100mg

Name: MedMol Trimipramine Maleate Salt 98% 100mg
Brand: MedMol
SKU: S85637-100mg

MedMol Trimipramine Maleate Salt 98% 100mg, complete specifications; suitable for production, research, laboratory testing and inspection; digital one-stop procurement platform for scientific materials.

item number：S85637-100mg

Product model：100mg

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Lead Time：30days

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MedMol Trimipramine Maleate Salt 98% 100mg

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