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Product details

名称

(-)-TK216

英文名称

(-)-TK216

货号

T655209-1ml

包装规格

1ml

浓度

10mM in DMSO

储存温度

-80℃储存

运输条件

超低温冰袋运输

产品介绍

(-)-TK216 is an enantiomer of TK216 . TK216 is an orally active and potent E26 transformation specific (ETS) inhibitor. (-)-TK216 has anti-cancer activity. In Vitro (-)-TK216 (compound 14; for 3 days) has an IC 50 In Vivo (-)-TK216 (compound 14; 5 mg/kg for iv or 25 mg/kg for po) has T 1/2 s of 0.8 hours and 3.1 hours, and AUCs of 4131 h•(ng/mL) and 13152 h•(ng/mL) for iv and po, respectively, in BALB/c mice or Sprague Dawley rats. MCE has not independently confirmed the accuracy of these methods. They are for reference only.

生化机理

(-)-TK216 是 TK216 ( HY-122903 ) 的对映体。TK216 是一种具有口服活性的强效 E26 转化特异性（ETS）抑制剂。(-)-TK216 具有抗癌活性。

CAS号

1903783-78-7(DMSO)

分子式

C19H15Cl2NO3

分子量

376.23 g/mol

Smiles

C1CC1C2=CC=C(C=C2)C(=O)CC3(C4=C(C=CC(=C4NC3=O)Cl)Cl)O

Safety

「No Dangerous Attributes」

「No upstream and downstream information yet」

Technical Documents

「No technical documents」

Articles

「No related articles yet」

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