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名称

TAK-683 acetate

别名

TAK-683醋酸盐

英文名称

TAK-683 acetate

货号

T658894-5mg

包装规格

5mg

浓度

≥98%

储存温度

避光,充氩,干燥,-80℃储存

运输条件

超低温冰袋运输

产品介绍

TAK-683 acetate is a potent full KISS1 receptor (KISS1R) agonist ( IC 50 =170 pM) with improved metabolic stability. TAK-683 acetate is a nonapeptide metastin analog, exhibits agonistic activities to KISS1R with EC 50 values of 0.96 nM and 1.6 nM for huma Appearance:Solid In Vitro:TAK-683 acetate exhibits an IC 50 value (95% CI) from receptor binding assays is 150-180 pM and EC 50 value (95% CI) from Ca + mobilization assays is 180 (159–203) pM in rat KISS1R-expressing Chinese hamster ovary (CHO) cells. MCE has not independent In Vivo:TAK-683 acetate (subcutaneous injection; 0.008, 0.08, 0.8, or 8 μmol/ml/kg; once daily; 7 days) induces an increase in plasma luteinizing hormone and testosterone levels; however, after day 7, plasma hormone levels and genital organ weights are reduced. Biological Activity:TAK-683 acetate is a potent full KISS1 receptor (KISS1R) agonist ( IC 50 =170 pM) with improved metabolic stability. TAK-683 acetate is a nonapeptide metastin analog, exhibits agonistic activities to KISS1R with EC 50 values of 0.96 nM and 1.6 nM for huma

分子式

C66H87N17O15

分子量

1358.5 g/mol

溶解性

H2O : 5 mg/mL (3.68 mM; Need ultrasonic)

Safety

「No Dangerous Attributes」

「No upstream and downstream information yet」

Technical Documents

「No technical documents」

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