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Product introduction

BI-3802 是一种高效的 BCL6 降解剂，能够抑制 BCL6 的Bric-à-brac (BTB) 结构域，IC50 值 ≤3 nM。BI-3802 可诱导 BCL6 蛋白聚集，并促进 E3 连接酶 SIAH1 介导的蛋白降解。BI-3802 具有抗肿瘤活性。 Information BI-3802 BI-3802 is a highly potent oncogenic transcription factor BCL6 degrader with strong de-repression of target genes anti-proliferative effects. BI-3802 inhibits the BTB domain of BCL6 with IC50 of ≤3 nM. BI-3802 exhibits antitumor activity. Targets BTB domain of BCL6 (Cell-free assay) 3 nM

Specs ⸢ View details ⸥

Chinese name

BI-3802, BCL6 转录抑制因子

English name

BI-3802

Chinese alias

English alias

Acetamide,2-[[6-[[5-chloro-2-[(3R,5S)-3,5-dimethyl-1-piperidinyl]-4-pyrimidinyl]amino]-1,2-dihydro-1-methyl-2-oxo-3-quinolinyl]oxy]-N-methyl-,rel-

CAS number

2166387-65-9

molecular formula

C24H29ClN6O3

molecular weight

484.98 g/mol

Exact mass

PSA

99.700 Å²

Logp

4.000

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