Share to

Overview

Specs

Technical Documents

Articles

reviews

Consult

returns

Product introduction

KZR-616（Zetomipzomib）是首创的免疫蛋白酶体 (immunoproteasome) 抑制剂，选择性靶向免疫蛋白酶体亚基 LMP7 (IC50: 39/57 nM=hLMP7/mLMP7) 和 LMP2 (IC50: 131/179 nM=hLMP7/mLMP7)。KZR-616用于多种自身免疫性疾病的潜力。 KZR-616（Zetomipzomib）, a first-in-class inhibitor of the immunoproteasome, selectively targets the LMP7 (IC50: 39/57 nM=hLMP7/mLMP7) and LMP2 (IC50: 131/179 nM=hLMP7/mLMP7) subunits of the immunoproteasome. KZR-616（Zetomipzomib）has the potential for the research of multiple autoimmune diseases.

Specs ⸢ View details ⸥

Chinese name

KZR-616, 蛋白酶体 20S 亚基 beta 2 抑制剂

English name

KZR-616

Chinese alias

English alias

(2S,3R)-N-((S)-3-(cyclopent-1-en-1-yl)-1-((R)-2-methyloxiran-2-yl)-1-oxopropan-2-yl)-3-hydroxy-3-(4-methoxyphenyl)-2-((S)-2-(2-morpholinoacetamido)propanamido)propanamide | BDBM50526811 | ZETOMIPZOMIB [INN] | D-Erythro-3-pentulose, 4,5-anhydro-1-(1-cyclop

CAS number

1629677-75-3

molecular formula

C30H42N4O8

molecular weight

586.68 g/mol

Exact mass

PSA

159.000 Å²

Logp

0.400

Technical Documents

「No technical documents」

「No upstream and downstream information yet」

Articles

「No related articles yet」

user reviews

Consultation

Warm reminder：

Because the manufacturer may temporarily adjust product specifications, prices, inventory, parameters and other information without notice, and there are differences in each user's consultation time and procurement needs, the platform reply content is only of reference value within a certain period. Sorry for the inconvenience caused to you, and thank you for your understanding and support! Please consult the online customer service for the latest details. Everything is subject to the real-time reply of the customer service.！

After Sales Services

Please check the quantity, appearance and product information in time when you receive the goods. In case of damage, wrong delivery, abnormal quality and other problems, please feel free to contact us.

Service Hotline:400-6226-992 ，We will handle it for you as soon as possible, thank you for your support and trust.！