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Product introduction

MDR-652是瞬时受体电位香草酸亚型 1 的选择性激动剂，对 hTRPV1 和 rTRPV1 的Ki 分别为 11.4 和 23.8 nM，EC50分别为 5.05 和 93 nM。MDR-652在缓解疼痛方面有研究的价值。 Information MDR-652 MDR-652 is a potent and specific agonist of transient receptor potential vanilloid 1 (TRPV1) with Ki of 11.4 nM and 23.8 nM for hTRPV1 and rTRPV1, respectively. MDR-652 has excellent and dose-dependent analgesic activity. Targets hTRPV1 (Cell-free assay); rTRPV1 (Cell-free assay) 11.4 nM(Ki); 23.8 nM(Ki)

Specs ⸢ View details ⸥

Chinese name

MDR-652

English name

MDR-652

Chinese alias

English alias

N-[[4-(3-chlorophenyl)-2-(1,1-dimethylethyl)-5-thiazolyl]methyl]-N'-[3-fluoro-4-(hydroxymethyl)phenyl]-urea

CAS number

1933528-96-1

molecular formula

C22H23ClFN3O2S

molecular weight

447.95 g/mol

Exact mass

≥97%

PSA

102.000 Å²

Logp

4.700

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